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1
DrugINNDate first registered by US FDACompany or CompaniesIndicationUS FDA Orphan indications (23-10-2020) (designations)CurrencyYears since 1st US FDA approvalCumulative revenue (in millions)202520242023202220212020201920182017201620152014201320122011201020092008200720062005200420032002200120001999199819971996199519941993199219911990
2
Kyproliscarfilzomib7/20/2012A generalCancer: Multiple Myeloma1USD12.8$1,960$562$554$467$306$71$0
3
Humiraadalimumab12/31/2002AbbvieRheumatoid arthritis (initial indication, now many more)9USD22.1$228,328$14,404$21,237$20,694$19,832$19,169$19,936$18,427$16,078$14,012$12,543$10,659$9,265$7,932$6,508$5,500$4,500$3,000$2,000$1,500$852$280$0
4
Humira (US only)adalimumab12/31/2002AbbvieRheumatoid arthritis (initial indication, now many more)9USD22.1$140,105$12,160$18,619$17,330$16,112$14,864$13,685$12,361$10,432$8,405$6,524$5,236$4,377
5
Humira (USA Medicare part B)adalimumab12/31/2002AbbvieRheumatoid arthritis (initial indication, now many more)9USD22.1$0
6
Humira (USA Medicare part D)adalimumab12/31/2002AbbvieRheumatoid arthritis (initial indication, now many more)9USD22.1$2,198
7
Viekiradasabuvir sodium; ombitasvir; paritaprevir; ritonavir12/19/2014AbbvieHCV1USD10.5$178$784$1,522$1,639$48
8
Viekira (US only)dasabuvir sodium; ombitasvir; paritaprevir; ritonavir12/19/2014AbbvieHCV1USD10.5$6$61$342$804$48
9
Viekira (USA Medicare Part B)dasabuvir sodium; ombitasvir; paritaprevir; ritonavir12/19/2014AbbvieHCV1USD10.5$0
10
Viekira (USA Medicare Part D)dasabuvir sodium; ombitasvir; paritaprevir; ritonavir12/19/2014AbbvieHCV1USD10.5$90$220
11
Ampyradalfampridine1/22/2010Acorda TherapeuticsMS2USD15.2$3,207$455$543$493$437$366$303$266$211$133
12
Ampyra (USA Medicare Part B)dalfampridine1/22/2010Acorda TherapeuticsMS2USD15.2$0
13
Ampyra (USA Medicare Part D)dalfampridine1/22/2010Acorda TherapeuticsMS2USD15.2$206$176$136$99$72
14
Soliriseculizumab paroxysmal nocturnal hemoglobinuria3/16/2007AlexionPNH; aHUS8USD18.0$28,981$1,874$4,064$3,946$3,563$3,144$2,843$2,591$2,234$1,551$1,134$783$541$387$259$66$0
15
Soliris (US only)eculizumab paroxysmal nocturnal hemoglobinuria3/16/2007AlexionPNH; aHUS8USD18.0$7,305$1,588$1,235$1,059$944$730$561$400$263$206$160$113$46$0
16
Soliris (USA Medicare part B)eculizumab paroxysmal nocturnal hemoglobinuria3/16/2007AlexionPNH; aHUS8USD18.0$267$233$178$142$98
17
Soliris (USA Medicare part D)eculizumab paroxysmal nocturnal hemoglobinuria3/16/2007AlexionPNH; aHUS8USD18.0$21$13$10$8$7
18
Teflaroceftaroline fosamil for injection10/29/2010
Allergan Sales (acquired Cerexa)
Acute skin infections, community-acquired pneumonia0USD14.5$577$128$122$134$138$56$0
19
Teflaro (USA Medicare Part B)ceftaroline fosamil for injection10/29/2010
Allergan Sales (acquired Cerexa)
Acute skin infections, community-acquired pneumonia0USD14.5$1$0.3$0.1$0.5$0.2
20
Teflaro (USA Medicare Part D)ceftaroline fosamil for injection10/29/2010
Allergan Sales (acquired Cerexa)
Acute skin infections, community-acquired pneumonia0USD14.5$12$10$7$4$2
21
Viibryd/Fetzimavilazodone1/21/2011
Allergan Sales (acquired Cerexa)
Mental illness: MDD0USD14.3$1,496$350$336$342$328$140$0
22
Viibryd/Fetzima (US only)vilazodone1/21/2011
Allergan Sales (acquired Cerexa)
Mental illness: MDD0USD14.3$342$333$342$328$140
23
Viibryd/Fetzima (USA Medicare Part B)vilazodone1/21/2011
Allergan Sales (acquired Cerexa)
Mental illness: MDD0USD14.3$0$0$0$0$0
24
Viibryd/Fetzima (USA Medicare Part D)vilazodone1/21/2011
Allergan Sales (acquired Cerexa)
Mental illness: MDD0USD14.3$74$66$57$42$22
25
Vascepaisocapent ethyl7/26/2012
Amarin Pharms (Amarin parent based in Ireland)
hypertriglyceridemia0EUR12.8
26
Enbreletanercept11/2/1998AmgenRheumatoid Arthritics; Plaque Psoriasis; Psoriaric Arthritics; Ankylosing Spondylitisl Juvenile Idiopathic Arthritis2USD26.2$26,464$5,014$5,433$5,965$5,364$4,688
27
Enbrel (US only)etanercept11/2/1998AmgenRheumatoid Arthritics; Plaque Psoriasis; Psoriaric Arthritics; Ankylosing Spondylitisl Juvenile Idiopathic Arthritis2USD26.2$25,235$4,807$5,206$5,719$5,099$4,404
28
Enbrel (USA Medicare part B)etanercept11/2/1998AmgenRheumatoid Arthritics; Plaque Psoriasis; Psoriaric Arthritics; Ankylosing Spondylitisl Juvenile Idiopathic Arthritis2USD26.2$0
29
Enbrel (USA Medicare part D)etanercept11/2/1998AmgenRheumatoid Arthritics; Plaque Psoriasis; Psoriaric Arthritics; Ankylosing Spondylitisl Juvenile Idiopathic Arthritis2USD26.2$1,572$1,385$1,198$977$722
30
Proliadenosumab6/1/2010AmgenOsteoperosis2USD14.9$9,688$2,291$1,968$1,635$1,312$1,030$744$472$203$33$0
31
Prolia (US only)denosumab6/1/2010AmgenOsteoperosis2USD14.9$1,500$1,272$1,049$837
32
Prolia (USA Medicare Part B)denosumab6/1/2010AmgenOsteoperosis2USD14.9$1,087$917$727$631$484
33
Prolia (USA Medicare Part D)denosumab6/1/2010AmgenOsteoperosis2USD14.9$185$151$114$73$38
34
Xgevadenosumab6/1/2010AmgenOsteoperosis2USD14.9$9,642$1,786$1,575$1,529$1,405$1,221$1,019$748$351$8$0
35
Xgeva (US only)denosumab6/1/2010AmgenOsteoperosis2USD14.9$1,338$1,157$1,115$1,006$857$764$644$343
36
Xgeva (USA Medicare Part B)denosumab6/1/2010AmgenOsteoperosis2USD14.9$0$0$0$0$0
37
Xgeva (USA Medicare Part D)denosumab6/1/2010AmgenOsteoperosis2USD14.9$15$12$9$6$4
38
Edarbiazilsartan kamedoxomil2/25/2011
Arbor Pharmaceuticals LLC
HTNEUR14.2
39
Horizantgabapentin enacarbil4/6/2011
Arbor Pharmaceuticals LLC
Restless Legs SyndromeEUR14.1
40
Xtandi (Astellas fiscal year)enzalutamide8/31/2012AstellasProstate cancer0JPY12.7Â¥3,137,200Â¥661,100Â¥534,300Â¥458,400Â¥400,000Â¥333,000Â¥294,300Â¥252,100Â¥137,200Â¥54,600Â¥12,200
41
Xtandi, USAenzalutamide8/31/2012AstellasProstate cancer0JPY12.7Â¥1,024,100Â¥276,900Â¥238,600Â¥203,500Â¥164,700Â¥140,400
42
Xtandi, Medicare (Federal fiscal year)enzalutamide8/31/2012AstellasProstate cancer0USD12.7$12,687$2,437$2,411$1,969$1,421$1,183$855$908$790.66$447$232$35
43
Xtandi, Medicaid (federal fiscal year)$132$116$98$72$53
44
Xtandi (Pfizer/Medivation alliance revenue)8/31/2012AstellasProstate cancer0USD12.7$3,291$1,198$1,185$1,024$838$699$590$140
45
Brilintaticagrelor7/20/2011AstraZenecaAcute coronary syndrome0USD13.8$4,727$1,321$1,079$839$619$476$283$89$21$0
46
Brilinta (US only)ticagrelor7/20/2011AstraZenecaAcute coronary syndrome0USD13.8$588$509$348$240$146$73$19$11
47
Brilinta (USA Medicare Part B)ticagrelor7/20/2011AstraZenecaAcute coronary syndrome0USD13.8$0$0$0$0$0
48
Brilinta (USA Medicare Part D)ticagrelor7/20/2011AstraZenecaAcute coronary syndrome0USD13.8$206$129$75$38$8
49
Tagrissoosimertinib11/13/2015AstraZenecaCancer: non-small-cell lung carcinomas 2USD9.6$3,257$1,860$955$423$19$0
50
Tagrisso (US only)osimertinib11/13/2015AstraZenecaCancer: non-small-cell lung carcinomas 2USD9.6$869$405$255
51
Tagrisso (USA Medicare part B)osimertinib11/13/2015AstraZenecaCancer: non-small-cell lung carcinomas 2USD9.6$0
52
Tagrisso (USA Medicare part D)osimertinib11/13/2015AstraZenecaCancer: non-small-cell lung carcinomas 2USD9.6$113
53
Xiaflexcollagenase clostridium histolyticum2/2/2010
Auxilium Pharmaceuticals (Acquired by Endo Pharmaceuticals)
Dupuytren's disease2USD15.2$826$265$213$190$158$0
54
Xiaflex (USA Medicare Part B)collagenase clostridium histolyticum2/2/2010
Auxilium Pharmaceuticals (Acquired by Endo Pharmaceuticals)
Dupuytren's disease2USD15.2$39$35$29$22$19.67
55
Xiaflex (USA Medicare Part D)collagenase clostridium histolyticum2/2/2010
Auxilium Pharmaceuticals (Acquired by Endo Pharmaceuticals)
Dupuytren's disease2USD15.2$3$2$2$1$0.80
56
Gadavistgadobutrol3/14/2011Bayer HealthcareCNS imagingEUR14.1€2,174€366€365€346€290€233€205€209€160€0
57
Gadavist (US only)gadobutrol3/14/2011Bayer HealthcareCNS imagingEUR14.1€112€116€104€86
58
Gadavist (USA Medicare Part B)gadobutrol3/14/2011Bayer HealthcareCNS imagingUSD14.1$5$4$3$2$2
59
Gadavist (USA Medicare Part D)gadobutrol3/14/2011Bayer HealthcareCNS imagingUSD14.1$0$0$0$0$0
60
Nataziaestradial valerate/dienogest tabs5/6/2010Bayer HealthcareFemale birth controlEUR15.0
61
Nexavarsorafenib12/1/2005Bayer HealthcareCancer: Hepatocellular carcinoma (HCC); renal cell carcinoma (RCC); thyroid carcinoma (DTC)5EUR19.3$8,540€712€834€870€892€773€771€792€725€705€604€462€270€130
62
Nexavar (US only)sorafenib12/1/2005Bayer HealthcareCancer: Hepatocellular carcinoma (HCC); renal cell carcinoma (RCC); thyroid carcinoma (DTC)5EUR19.3$1,146€216€294€312€324
63
Nexavar (USA Medicare part B)sorafenib12/1/2005Bayer HealthcareCancer: Hepatocellular carcinoma (HCC); renal cell carcinoma (RCC); thyroid carcinoma (DTC)5USD19.3$0$0$0$0$0
64
Nexavar (USA Medicare part D)sorafenib12/1/2005Bayer HealthcareCancer: Hepatocellular carcinoma (HCC); renal cell carcinoma (RCC); thyroid carcinoma (DTC)5USD19.3$844$214$206$169$138$117
65
Stivargaregorafenib9/27/2012Bayer HealthcareCancer: GISTEUR12.6€315€315€275€313€224€197
66
Stivarga (US only)regorafenib9/27/2012Bayer HealthcareCancer: GISTEUR12.6€149€166€142€181
67
Stivarga (USA Medicare Part B)regorafenib9/27/2012Bayer HealthcareCancer: GISTUSD12.6$0$0$0$0$0
68
Stivarga (USA Medicare Part D)regorafenib9/27/2012Bayer HealthcareCancer: GISTUSD12.6$76$100$87$84$12
69
Avonexinterferon beta-1a5/17/1996BiogenMSUSD28.6$34,350$1,916$2,152$2,314$2,630$3,013$3,006$2,913$2,687$2,518$2,323$2,203$1,868$1,707$1,543$1,417$143
70
Avonex (US only)interferon beta-1a5/17/1996BiogenMSUSD28.6$1,420$1,594$1,675$1,790$1,957$1,902$1,794
71
Avonex (USA Medicare Part B)interferon beta-1a5/17/1996BiogenMSUSD28.6$5$4$6
72
Avonex (USA Medicare Part D)interferon beta-1a5/17/1996BiogenMSUSD28.6$295$312$326$367$390
73
Spinrazanusinersen12/23/2016BiogenSpinal muscular atrophy (SMA)1USD8.5$4,710$2,097$1,724$884$5
74
Spinraza (US only)nusinersen12/23/2016BiogenSpinal muscular atrophy (SMA)1USD8.5$854$657$5
75
Spinraza (USA Medicare Part B)nusinersen12/23/2016BiogenSpinal muscular atrophy (SMA)1USD8.5$0
76
Spinraza (USA Medicare Part D)nusinersen12/23/2016BiogenSpinal muscular atrophy (SMA)1USD8.5$0
77
Tecfideradimethyl fumarate3/27/2013Biogen IDECMS0USD12.1$19,880$4,274$4,214$3,968$3,638$2,909$876
78
Tecfidera (US only)dimethyl fumarate3/27/2013Biogen IDECMS0USD12.1$3,294$3,169$2,908$2,427$864
79
Tecfidera (USA Medicare part B)dimethyl fumarate3/27/2013Biogen IDECMS0USD12.1$0$0$0$0
80
Tecfidera (USA Medicare part D)dimethyl fumarate3/27/2013Biogen IDECMS0USD12.1$932$876$599$159
81
Opdivonivolumab12/22/2014BMSCancer: NSCLC11USD10.5$23,609$7,204$6,735$4,948$3,774$942$6$0
82
Opdivo (US only)nivolumab12/22/2014BMSCancer: NSCLC11USD10.5$15,173$4,344$4,239$3,102$2,664$823$1
83
Opdivo (USA Medicare Part B)nivolumab12/22/2014BMSCancer: NSCLC11USD10.5$0$0
84
Opdivo (USA Medicare Part D)nivolumab12/22/2014BMSCancer: NSCLC11USD10.5$26$11
85
Pradaxadabigatran etexilate mesylate10/19/2010Boehringer Ingelheim Stroke0EUR14.5€6,8751,3851,2871,1981,2061,108$629$62$0
86
Pradaxa (USA Medicare Part B)dabigatran etexilate mesylate10/19/2010Boehringer Ingelheim Stroke0USD14.5$0$0$0$0$0
87
Pradaxa (USA Medicare Part D)dabigatran etexilate mesylate10/19/2010Boehringer Ingelheim Stroke0USD14.5$607$570$557$500$391
88
SpirivaTiotropium Bromide1/30/2004Boehringer Ingelheim COPD1EUR21.1€2,826€2,995€3,553€3,237€3,552€3,562€3,153
89
Spiriva (US only)Tiotropium Bromide1/30/2004Boehringer Ingelheim COPD1USD21.1$1,865
90
Spiriva (USA Medicare Part B)Tiotropium Bromide1/30/2004Boehringer Ingelheim COPD1USD21.1$0$0$0$0$0
91
Spiriva (USA Medicare Part D)Tiotropium Bromide1/30/2004Boehringer Ingelheim COPD1USD21.1$1,819$2,191$2,158$1,959$1,603
92
Tradjentalinagliptin5/2/2011Boehringer Ingelheim Diabetes0EUR14.0€4,0061,3331,128$909$636$0
93
Tradjenta (USA Medicare part B)linagliptin5/2/2011Boehringer Ingelheim Diabetes0USD$0
94
Tradjenta (USA Medicare part D)linagliptin5/2/2011Boehringer Ingelheim Diabetes0USD14.0$708$508$292$153$35
95
Daklinzadaclatasvir dihydrochloride7/24/2015
Bristol-Myers Squibb (BMS)
HCVUSD9.9$386$1,550$1,315
96
Daklinza (USA Medicare Part B)daclatasvir dihydrochloride7/24/2015
Bristol-Myers Squibb (BMS)
HCVUSD9.9$0
97
Daklinza (USA Medicare Part D)daclatasvir dihydrochloride7/24/2015
Bristol-Myers Squibb (BMS)
HCVUSD9.9$391$112
98
Eliquisapixaban12/28/2012
Bristol-Myers Squibb (BMS)
Heart Disease: Stroke0USD12.4$7,929$6,438
99
Spryceldasatinib6/28/2006
Bristol-Myers Squibb (BMS)
Cancer: Chronic Myeloid Leukemia (CML)4USD18.7$15,644$2,110$2,000$2,005$1,824$1,620$1,493$1,280$1,019$803$576$421$310$158$25$0
100
Sprycel (US only)dasatinib6/28/2006
Bristol-Myers Squibb (BMS)
Cancer: Chronic Myeloid Leukemia (CML)4USD18.7$1,091$1,105$969$829$671$541$404$294$188$123$92$58