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1 | Callaix.com List of Medicines | from https://callaix.com/medicines | ||||||||||||||||||||||||
2 | ||||||||||||||||||||||||||
3 | Medicine | Trade Name | Category | Sub-category 1 | Sub-category 2 | Year of First FDA approval | Types of Cancer | |||||||||||||||||||
4 | Abemaciclib | Verzenio | Kinase Inhibitor | CDK (Cyclin-Dependent Kinase) Inhibitor | 2017 | breast cancer | ||||||||||||||||||||
5 | Abiraterone | Zytiga | Anti-Androgen | CYP17A1 inhibitor | 2011 | prostate cancer | ||||||||||||||||||||
6 | Acalabrutinib | Calquence | Kinase Inhibitor | BTK inhibitor | 2017 | mantle cell carcinoma, chronic lymphocytic leukemia | ||||||||||||||||||||
7 | Actinomycin-D | Act-D, Cosmegen, Dactinomycin | Antibiotic | 1964 | many sarcomas and some carcinomas | |||||||||||||||||||||
8 | Ado-trastuzumab | Kadcyla | Antibody-drug conjugate | HER2 inhibitor | 2019 | breast cancer | ||||||||||||||||||||
9 | Afatinib | Gilotrif | Kinase Inhibitor | 2013 | non-small cell lung cancer | |||||||||||||||||||||
10 | Aldesleukin | Proleukin | Immunostimulant | 1992 | melanoma, renal cell carcinoma | |||||||||||||||||||||
11 | Alectinib | Alecensa | Kinase Inhibitor | 2015 | non-small cell lung cancer | |||||||||||||||||||||
12 | Alemtuzumab | Campath | Monoclonal Antibody | 2014 | B-cell chronic lymphocytic leukemia | |||||||||||||||||||||
13 | Alpelisib | Piqray | PI3K Inhibitor | 2019 | breast cancer | |||||||||||||||||||||
14 | Alitretinoin | Panretin, Toctino | Retinoid | 1999 | Karposi's sarcoma | |||||||||||||||||||||
15 | Altretamine | Hexalen | Alkylating agent | 1990 | ovarian cancer | |||||||||||||||||||||
16 | Amivantamab-vmjw | Rybrevant | Monoclonal Antibody | 2021 | non-small cell lung cancer | |||||||||||||||||||||
17 | Aminoglutethimide | Cytadren | Aromatase inhibitor | 1980 | breast cancer, prostate cancer | |||||||||||||||||||||
18 | Anastrozole | Arimidex | Aromatase inhibitor | 1995 | breast cancer | |||||||||||||||||||||
19 | Apalutamide | Erleada | Anti-Androgen | 2019 | prostate cancer | |||||||||||||||||||||
20 | Arsenic Trioxide | Other | 2000 | leukemia | ||||||||||||||||||||||
21 | Asciminib | Scemblix | Kinase Inhibitor | 2021 | leukemia | |||||||||||||||||||||
22 | Asparaginase, L-asparaginase | Elspar, Kidrolase | Enzyme | 2011 | acute lymphocytic leukemia | |||||||||||||||||||||
23 | Atezolizumab | Tecentriq | Monoclonal Antibody | checkpoint inhibitor | Anti-PD-1 | 2016 | small cell lung cancer, urothelial carcinoma, breast cancer, non-small cell lung cancer | |||||||||||||||||||
24 | Avapritinib | Ayvakit | Kinase Inhibitor | 2020 | gastrointestinal stromal tumor | |||||||||||||||||||||
25 | Avelumab | Bavencio | Monoclonal Antibody | checkpoint inhibitor | Anti-PD-1 | 2017 | merkel cell carcinoma, renal cell carcinoma, urothelial carcinoma | |||||||||||||||||||
26 | Axicabtagene | Yescarta | CAR T-Cell therapy | 2017 | lymphoma | |||||||||||||||||||||
27 | Axitinib | Inlyta | Kinase Inhibitor | VEGF/VEGFR inhibitor | 2012 | renal cell carcinoma | ||||||||||||||||||||
28 | Azacitidine | Vidaza | Antimetabolite | 2004 | myelodysplastic syndromes, leukemia | |||||||||||||||||||||
29 | Belantamab mafodotin-blmf | Blenrep | Monoclonal Antibody | 2020 | multiple myeloma | |||||||||||||||||||||
30 | Belinostat | Beleodaq | HDAC Inhibitor | 2014 | lymphoma | |||||||||||||||||||||
31 | Bendamustine | Treanda | Alkylating Agent | Mustard | 2008 | B-cell non-Hodgkin lymphoma, Chronic lymphocytic leukemia | ||||||||||||||||||||
32 | Bevacizumab | Avastin | Monoclonal Antibody | Angiogenesis inhibitor | VEGF/VEGFR inhibitor | 2004 | colorectal cancer, renal cell carcinoma, cervical cancer, glioblastoma, nonsquamous non-small cell lung cancer, ovarian epithelial cancer | |||||||||||||||||||
33 | Bexarotene | Targretin | Retinoid | 1999 | Skin problems caused by cutaneous T-cell lymphoma | |||||||||||||||||||||
34 | Bicalutamide | Casodex | Anti-Androgen | 1995 | prostate cancer | |||||||||||||||||||||
35 | Binimetinib | Mektovi | Kinase Inhibitor | 2018 | melanoma | |||||||||||||||||||||
36 | Bleomycin | Blenoxane | Antibiotic | 1979 | lymphoma, melanoma, sarcoma, ovarian cancer, testicular cancer | |||||||||||||||||||||
37 | Blinatumomab | Blincyto | Monoclonal Antibody | 2014 | B-cell acute lymphoblastic leukemia | |||||||||||||||||||||
38 | Bortezomib | Velcade | Proteasome inhibitor | 2003 | mantle cell lymphoma, multiple myeloma | |||||||||||||||||||||
39 | Bosutinib | Bosulif | Kinase Inhibitor | Bcr-Abl inhibitor | 2012 | chronic myelogenous leukemia | ||||||||||||||||||||
40 | Brentuximab vedotin | Adcetris | Antibody-drug conjugate | 2011 | peripheral T-cell lymphoma, cutaneous T-cell lymphoma, cutaneous anaplastic large cell lymphoma, Hodgkin's Disease, anaplastic large cell lymphoma | |||||||||||||||||||||
41 | Brigatinib | Alunbrig | Kinase Inhibitor | ALK inhibitor | 2017 | non-small cell lung cancer | ||||||||||||||||||||
42 | Busulfan | Myleran | Alkylating Agent | Alkyl sulfonate | 1999 | chronic myelogenous leukemia | ||||||||||||||||||||
43 | Cabazitaxel | Jevtana | Mitotic Inhibitor | Taxane | 2010 | prostate cancer | ||||||||||||||||||||
44 | Cabozantinib | Cabometyx | Kinase Inhibitor | VEGF/VEGFR inhibitor | 2012 | renal cell carcinoma, hepatocellular carcinoma, medullary thyroid cancer | ||||||||||||||||||||
45 | Calaspargase pegol-mknl | Asparlas | Enzyme | 2018 | acute lymphoblastic leukemia | |||||||||||||||||||||
46 | Camptothecin | Camptosar | Topoisomerase inhibitor | 2012 | colon cancer, rectal cancer | |||||||||||||||||||||
47 | Capecitabine | Xeloda | Antimetabolite | Prodrug of Fluorouracil | 2005 | Breast cancer, colorectal cancer | ||||||||||||||||||||
48 | Capmatinib | Tabrecta | Kinase Inhibitor | 2020 | non small-cell lung cancer | |||||||||||||||||||||
49 | Carboplatin | Paraplatin | Alkylating Agent | Platinum compound | 1989 | ovarian cancer and other types | ||||||||||||||||||||
50 | Carfilzomib | Kyprolis | Proteasome inhibitor | 2012 | multiple myeloma | |||||||||||||||||||||
51 | Carmustine | BiCNU | Alkylating Agent | Nitrosurea | 1996 | brain tumors, Hodgkin's Disease, multiple myeloma, Non-Hodgkin's lymphoma | ||||||||||||||||||||
52 | Cemiplimab-rwlc | Libtayo | Monoclonal Antibody | checkpoint inhibitor | Anti-PD-1 | 2018 | cutaneous squamous cell carcinoma | |||||||||||||||||||
53 | Ceritinib | Zykadia | Kinase Inhibitor | ALK inhibitor | 2014 | non-small cell lung cancer | ||||||||||||||||||||
54 | Cetuximab | Erbitux | Monoclonal Antibody | EGFR inhibitor | 2009 | colorectal cancer, squamous cell carcinoma of the head and neck, non-small cell lung cancer | ||||||||||||||||||||
55 | Clofarabine | Clolar | antimetabolite | 2014 | acute lymphoblastic leukemia | |||||||||||||||||||||
56 | Chlorambucil | Leukeran | Alkylating Agent | Mustard | 1957 | Chronic lymphocytic leukemia, Hodgkin's disease. Non-Hodgkin's lymphoma, ovarian cancer, testicular cancer, and others | ||||||||||||||||||||
57 | Cisplatin | Platinol | Alkylating Agent | Platinum compound | 1978 | bladder cancer, testicular cancer, ovarian cancer, esophageal, lung, breast, cervical, stomach and prostate cancers | ||||||||||||||||||||
58 | Cladribine | Litak and Movectro | Antimetabolite | Adenosine deaminase inhibitor | 1993 | hairy cell leukemia, acute myeloid leukemia, chronic lymphocytic leukemia, lymphoma | ||||||||||||||||||||
59 | Cobimetinib | Cotellic | MEK Inhibitor | 2015 | melanoma | |||||||||||||||||||||
60 | Copanlisib | Aliqopa | PI3K Inhibitor | 2017 | follicular lymphoma | |||||||||||||||||||||
61 | Crizotinib | Xalkori | Kinase Inhibitor | 2011 | non-small cell lung cancer | |||||||||||||||||||||
62 | Cyclophosphamide | Endoxan, Cytoxan, Neosar | Alkylating Agent | Mustard | 1959 | Retinoblastoma, Chronic myelogenous leukemia, Hodgkin's disease, Multiple myeloma, Mycosis fungoides, Neuroblastoma, Non-Hodgkin lymphoma, Acute lymphoblastic leukemia, Acute monocytic leukemia, Acute myeloid leukemia, Breast cancer, Chronic granulocytic leukemia. Chronic lymphocytic leukemia | ||||||||||||||||||||
63 | Cytarabine | Cytosar-U, Arabinosylcytosine | Antimetabolite | 1969 | Acute lymphoblastic leukemia (ALL), Acute myeloid leukemia (AML), Chronic myelogenous leukemia (CML), promyelocytic leukemia | |||||||||||||||||||||
64 | Dabrafenib | Taflinar | Kinase Inhibitor | BRAF inhibitor | 2013 | anaplastic thyroid cancer, melanoma, non-small cell lung cancer | ||||||||||||||||||||
65 | Dacarbazine | DTIC, DTIC-Dome | Alkylating Agent | 1975 | melanoma, Hodgkin's Disease, sarcomas, neuroblastoma, and thyroid cancer | |||||||||||||||||||||
66 | Dacomitinib | Vizimpro | Kinase Inhibitor | EGFR inhibitor | HER2 inhibitor | 2018 | non-small cell lung cancer | |||||||||||||||||||
67 | Daratumumab | Darzalex | Monoclonal Antibody | 2015 | multiple myeloma | |||||||||||||||||||||
68 | Darolutamide | Nubeqa | Anti-Androgen | 2019 | prostate cancer | |||||||||||||||||||||
69 | Dasatinib | Sprycel | Kinase Inhibitor | Bcr-Abl inhibitor | 2006 | acute myeloid leukemia, chronic lymphocytic leukemia | ||||||||||||||||||||
70 | Daunorubicin | DaunoXome, Cerubidine | Anthracycline | Antibiotic | 1979 | acute lymphoblastic leukemia, acute myelogenous leukemia, acute promyelocytic leukemia | ||||||||||||||||||||
71 | Decitabine | Dacogen | Antimetabolite | Cytosine Analog | 2006 | Myelodysplastic syndromes | ||||||||||||||||||||
72 | Degarelix | Firmagon | Anti-Androgen | 2008 | prostate cancer | |||||||||||||||||||||
73 | Denileukin diftitox | Ontak | Antibody-drug conjugate | no longer on market | 1999 | leukemia and lymphoma | ||||||||||||||||||||
74 | Dinutuximab | Unituxin | Monoclonal Antibody | 2015 | neuroblastoma | |||||||||||||||||||||
75 | Docetaxel | Taxotere | Mitotic Inhibitor | taxane | 1996 | breast, prostate, stomach cancer, non-small cell lung cancer, head and neck cancer | ||||||||||||||||||||
76 | Dostarlimab-gxly | Jemperli | Monoclonal Antibody | 2021 | endometrial cancer | |||||||||||||||||||||
77 | Doxorubicin | Adriamycin | Anthracycline | Antibiotic | 1974 | lymphoblastic and myeloid leukemia, breast cancer, stomach cancer, Hodgkin's lymphoma, neuroblastoma, non-Hodgkin lymphoma, ovarian cancer, small cell lung cancer, soft tissue and bone sarcomas, thyroid cancer, bladder cancer, Wilms tumor. | ||||||||||||||||||||
78 | Durvalumab | Imfinzi | Monoclonal Antibody | checkpoint inhibitor | Anti-PD-1 | 2017 | non-small cell lung cancer, urothelial carcinoma | |||||||||||||||||||
79 | Duvelisib | Copiktra | PI3K Inhibitor | 2018 | follicular lymphoma, chronic lymphocytic leukemia, small lymphocytic lymphoma | |||||||||||||||||||||
80 | Elotuzumab | Emplicit | Monoclonal Antibody | 2015 | multiple myeloma | |||||||||||||||||||||
81 | Enasidenib | Idhifa | IDH2 inhibitor | 2017 | acute myeloid leukemia | |||||||||||||||||||||
82 | Encorafenib | Braftovi | Kinase Inhibitor | BRAF inhibitor | 2018 | melanoma | ||||||||||||||||||||
83 | Enfortumab vedotin-ejfv | Padcev | Antibody-drug conjugate | 2019 | urothelial cancer | |||||||||||||||||||||
84 | Entrectinib | Rozlytrek | Kinase Inhibitor | 2019 | non-small cell lung cancer | |||||||||||||||||||||
85 | Enzalutamide | Xtandi | Anti-androgen | 2012 | prostate cancer | |||||||||||||||||||||
86 | Epirubicin | Ellence | Anthracycline | Antibiotic | 1999 | breast cancer | ||||||||||||||||||||
87 | Erdafitinib | Balversa | Kinase Inhibitor | FGFR inhibitor | 2019 | urothelial carcinoma and bladder cancer | ||||||||||||||||||||
88 | Eribulin | Halaven | Mitotic Inhibitor | 2010 | breast cancer | |||||||||||||||||||||
89 | Erlotinib | Tarceva | Kinase Inhibitor | EGFR inhibitor | 2004 | pancreatic cancer, non-smell lung cancer | ||||||||||||||||||||
90 | Estramustine | Emcyt, Estracit | Hormone Suppressant | Mustard | 1981 | prostate cancer | ||||||||||||||||||||
91 | Etoposide | Eposin, Vepesid | Topoisomerase inhibitor | plant alkaloid | 1983 | small cell lung cancer, testicular cancer | ||||||||||||||||||||
92 | Everolimus | Afinitor, Zortress | mTOR inhibitor | 2010 | kidney, breast, pancreatic, gastrointestinal, lung cancer, sarcomas, lymphomas | |||||||||||||||||||||
93 | Exemestane | Aromasin | Aromatase Inhibitor | 1999 | breast cancer | |||||||||||||||||||||
94 | Fam-trastuzumab deruxtecan-nxki | Enhertu | Antibody-drug conjugate | 2019 | breast cancer | |||||||||||||||||||||
95 | Fluorouracil (5-FU) | Adrucil | Antimetabolite | 1962 | bladder, anal, breast, gastrointestinal, thymic, cervical, head and neck, and colorectal cancer | |||||||||||||||||||||
96 | Floxuridine | FUDR | Antimetabolite | pyrimidine analog | 1970 | stomach, colon, kidney cancer | ||||||||||||||||||||
97 | Fludarabine | Fludara | Antimetabolite | purine analog | 1991 | lymphocytic leukemia, non-Hodgkins lymphoma | ||||||||||||||||||||
98 | Flutamide | Eulexin | Anti-androgen | 1989 | prostate cancer | |||||||||||||||||||||
99 | Fulvestrant | Faslodex | Anti-androgen | 2002 | breast cancer | |||||||||||||||||||||
100 | Gefitinib | Iressa | Kinase Inhibitor | EGFR inhibitor | 2003 | non-small cell lung cancer |