A | B | C | D | E | F | G | H | I | J | K | L | M | N | O | P | Q | R | S | T | U | V | W | X | Y | Z | AA | AB | AC | AD | AE | AF | AG | AH | AI | AJ | AK | AL | AM | AN | AO | AP | AQ | AR | AS | AT | AU | AV | AW | AX | AY | AZ | BA | BB | |
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1 | OSA No. | Salt | Batch | Target | Target % activity | SMILES_parent | Img | Name | InChiKey | VendorID/ LabNotebook ID/Other Code | MW_parent | Fragalysis_ref | Source | Status | Wiki link | MountingResult | DataCollectionOutcome | LigandBound | ChEMBL | Drugbank | PDBligand | Guide to Pharm | Drugs of the Future | Kegg Ligand | ChEBI | NIH Clinical | ZINC | eMolecules | IBM IP | Gene Expression | NFDA Substance | SureChEMBL Patents | PharmGKB | Human Metab | Selleck | Thomson Pharma | Pubchem | Mcule | NMR shift DB | Networks | Toxicology Resource | MolPort | Japanese Chemicals | BindingDB | CompTox | Lipidmaps | DrugCentral | Carotenoid | Metabolights | Brenda | rhea | chemicalbook | swisslipids | gsrs |
12 | OSA_001041 | XX | 01 | MurC | CN1C(N)=CC(C(C)(C)C)=N1 | 3-(tert-butyl)-1-methyl-1H-pyrazol-5-amine | XSCDSAMVQLKDNI-UHFFFAOYSA-N | WYH5-X-P | 153.23 | |||||||||||||||||||||||||||||||||||||||||||||
13 | OSA_001042 | XX | 01 | MurC | CC(C)(C)C1=NN(C)C(NC(NC2=CC=C(Cl)C=C2)=O)=C1 | 1-(3-(tert-butyl)-1-methyl-1H-pyrazol-5-yl)-3-(4-chlorophenyl)urea | FWIJKWMXNHRSRO-UHFFFAOYSA-N | WYH6-X-P | 306.79 | |||||||||||||||||||||||||||||||||||||||||||||
14 | OSA_001043 | XX | 01 | MurC | ClC1=NC2=C(C=NN2)C(NC3=NNC(C(C)C)=C3)=N1 | 6-chloro-N-(5-isopropyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | SIOMWOBKQAVWMK-UHFFFAOYSA-N | WYH8-X-P | 277.72 | |||||||||||||||||||||||||||||||||||||||||||||
15 | OSA_001044 | XX | 01 | MurC | CC(C)C1=CC(NC2=NC(N[C@@H](CO)C3CCCCC3)=NC4=C2C=NN4)=NN1 | (R)-2-cyclohexyl-2-((4-((5-isopropyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)ethan-1-ol | ISQKTZJQIVTQSH-HNNXBMFYSA-N | WYH9-X-P | 384.49 | |||||||||||||||||||||||||||||||||||||||||||||
16 | OSA_001045 | XX | 01 | MurC | CC(C)(C)C1=CC(N2C(C)=CC=C2C)=NN1 | 5-(tert-butyl)-3-(2,5-dimethyl-1H-pyrrol-1-yl)-1H-pyrazole | OEMSXMRZOUJFOH-UHFFFAOYSA-N | WYH11-X-P | 217.32 | |||||||||||||||||||||||||||||||||||||||||||||
17 | OSA_001046 | XX | 01 | MurC | CC(C)(C)C1=NN(C)C(N2C(C)=CC=C2C)=C1 | 3-(tert-butyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-1-methyl-1H-pyrazole | GJEZAWGSKCLSGW-UHFFFAOYSA-N | WYH12-X-P1 | 231.34 | |||||||||||||||||||||||||||||||||||||||||||||
18 | OSA_001047 | XX | 01 | MurC | CC(C)(C)C1=CC(N2C(C)=CC=C2C)=NN1C | 5-(tert-butyl)-3-(2,5-dimethyl-1H-pyrrol-1-yl)-1-methyl-1H-pyrazole | TZHZITZMYWTHSP-UHFFFAOYSA-N | WYH12-X-P2 | 231.34 | |||||||||||||||||||||||||||||||||||||||||||||
19 | OSA_001048 | XX | 01 | MurC | CN1C(C(C)(C)C)=CC(N)=N1 | 5-(tert-butyl)-1-methyl-1H-pyrazol-3-amine | KYZWYUQUBBZLPO-UHFFFAOYSA-N | WYH13-X-P | 153.23 | |||||||||||||||||||||||||||||||||||||||||||||
20 | OSA_001049 | XX | 01 | MurC | CC(C)(C)C1=CC(NC(NC2=CC=C(Cl)C=C2)=O)=NN1C | 1-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-3-(4-chlorophenyl)urea | PSTXVVILKIZARC-UHFFFAOYSA-N | WYH15-X-P | 306.79 | |||||||||||||||||||||||||||||||||||||||||||||
21 | OSA_001050 | XX | 01 | MurC | CN1C(C(C)(C)C)=CC(NC2=NC(Cl)=NC3=C2C=NN3)=N1 | N-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-6-chloro-1H-pyrazolo[3,4-d]pyrimidin-4-amine | FODXCYLKXVFESG-UHFFFAOYSA-N | WYH16-X-P | 305.77 | |||||||||||||||||||||||||||||||||||||||||||||
22 | OSA_001051 | XX | 01 | MurC | CC(C)(C)C1=CC(NC2=NC(N[C@H](CO)C3=CC=CC=C3)=NC4=C2C=NN4)=NN1C | (S)-2-((4-((5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)-2-phenylethan-1-ol | MOLGZLFXZJMRCB-OAHLLOKOSA-N | WYH17-X-P | 406.49 | |||||||||||||||||||||||||||||||||||||||||||||
23 | OSA_001071 | XX | 01 | MurC | OC[C@H](NC1=NC2=C(C=NN2)C(NC3=NN(C)C(C(C)(C)C)=C3)=N1)C4=CC=CC=C4 | (R)-2-((4-((5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)-2-phenylethan-1-ol | MOLGZLFXZJMRCB-HNNXBMFYSA-N | WYH25-1-P | 406.49 | |||||||||||||||||||||||||||||||||||||||||||||
24 | OSA_001095 | xx | 01 | MurC | NC[C@H](NC1=NC2=C(C=NN2)C(NC3=NN(C)C(C(C)(C)C)=C3)=N1)C4=CC=CC=C4 | (R)-N6-(2-amino-1-phenylethyl)-N4-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | DINXXNJQQKPNGS-HNNXBMFYSA-N | WYH22-1-P | 405.51 | |||||||||||||||||||||||||||||||||||||||||||||
25 | OSA_001095 | xx | 02 | MurC | NC[C@H](NC1=NC2=C(C=NN2)C(NC3=NN(C)C(C(C)(C)C)=C3)=N1)C4=CC=CC=C4 | (R)-N6-(2-amino-1-phenylethyl)-N4-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | DINXXNJQQKPNGS-HNNXBMFYSA-N | WYH22-2-P | 405.51 | |||||||||||||||||||||||||||||||||||||||||||||
26 | OSA_001111 | XX | 01 | MurC | CC(C)(C)C1=CC(NC2=C3C(NN=C3)=NC(N[C@@H](CC4)CC[C@H]4N)=N2)=NN1C | N6-((1r,4r)-4-aminocyclohexyl)-N4-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | PGFATVWGNSDBAF-HAQNSBGRSA-N | WYH30-1-P | 383.5 | |||||||||||||||||||||||||||||||||||||||||||||
27 | OSA_001112 | XX | 01 | MurC | CC(C)(C)C1=CC(NC2=C3C(NN=C3)=NC(NCCOCCOCCN)=N2)=NN1C | N6-(2-(2-(2-aminoethoxy)ethoxy)ethyl)-N4-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | GYAFMGRTCRSKGQ-UHFFFAOYSA-N | WYH32-1-P | 417.52 | |||||||||||||||||||||||||||||||||||||||||||||
28 | OSA_001174 | FA | 01 | MurC | CC(C)(C)C1=CC(NC2=NC(NC3CCC(NC(N)=N)CC3)=NC4=C2C=NN4)=NN1C | 1-(4-((4-((5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)cyclohexyl)guanidine | COHCMYHZVFQCSM-UHFFFAOYSA-N | WYH76-1-P (WYH30-G) | 425.5 | |||||||||||||||||||||||||||||||||||||||||||||
29 | OSA_001175 | XX | 01 | MurC | CC(C)(C)C1=CC(NC2=NC(N[C@H]3[C@H](O)CC4=CC=CC=C43)=NC5=C2C=NN5)=NN1C | (1R,2R)-1-((4-((5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)-2,3-dihydro-1H-inden-2-ol | OTFLFRAEUDDJKT-CRAIPNDOSA-N | WYH77-1-P | 418.5 | |||||||||||||||||||||||||||||||||||||||||||||
30 | OSA_001176 | XX | 01 | MurC | CC(C)(C)C1=CC(NC2=NC(N[C@H]3[C@@H](O)CC4=CC=CC=C43)=NC5=C2C=NN5)=NN1C | (1R,2S)-1-((4-((5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)-2,3-dihydro-1H-inden-2-ol | OTFLFRAEUDDJKT-MAUKXSAKSA-N | WYH78-1-P | 418.5 | |||||||||||||||||||||||||||||||||||||||||||||
31 | OSA_001177 | FA | 01 | MurC | CC(C)(C)C1=CC(NC2=NC(N[C@H]3CC4=C(C=CC=C4)[C@@H]3N)=NC5=C2C=NN5)=NN1C | N6-((1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl)-N4-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | XSKJBNCXGBWYOO-YJBOKZPZSA-N | WYH85-2-P | 417.5 | |||||||||||||||||||||||||||||||||||||||||||||
32 | OSA_001178 | FA | 01 | MurC | CC(C)(C)C1=CC(NC2=NC(N[C@@H]3CC4=C(C=CC=C4)[C@H]3N)=NC5=C2C=NN5)=NN1C | N6-((1R,2R)-1-amino-2,3-dihydro-1H-inden-2-yl)-N4-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | XSKJBNCXGBWYOO-CRAIPNDOSA-N | WYH86-2-P | 417.5 | |||||||||||||||||||||||||||||||||||||||||||||
33 | OSA_001179 | FA | 01 | MurC | WYH87-1-P | 459.6 | ||||||||||||||||||||||||||||||||||||||||||||||||
34 | OSA_001180 | FA | 01 | MurC | CC(C)(C)C1=CC(NC2=NC(N[C@@H]3CC4=C(C=CC=C4)[C@H]3NC(N)=N)=NC5=C2C=NN5)=NN1C | 1-((1R,2R)-2-((4-((5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)-2,3-dihydro-1H-inden-1-yl)guanidine | JHDIHLQPZRBFCN-CRAIPNDOSA-N | WYH88-1-P | 459.6 | |||||||||||||||||||||||||||||||||||||||||||||
35 | OSA_001181 | XX | 01 | MurC | WYH23/24-X-P | |||||||||||||||||||||||||||||||||||||||||||||||||
36 | OSA_001182 | XX | 01 | MurC | WYH54-X-P | |||||||||||||||||||||||||||||||||||||||||||||||||
37 | OSA_001183 | XX | 01 | MurC | WYH62-X-P | |||||||||||||||||||||||||||||||||||||||||||||||||
38 | OSA_001184 | XX | 01 | MurC | WYH61-X-P | |||||||||||||||||||||||||||||||||||||||||||||||||
39 | OSA_001201 | XX | 01 | MurC | NC1=NC(NC2=NNC(C(C)(C)C)=C2)=C3C(NN=C3)=N1 | N4-(5-(tert-butyl)-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | WQXHYTAUJLYLSF-UHFFFAOYSA-N | WYH_TR1-4-1-P | 272.3 | |||||||||||||||||||||||||||||||||||||||||||||
40 | OSA_001202 | XX | 01 | MurC | WYH22-R-Boc (WYH21-R-P) | |||||||||||||||||||||||||||||||||||||||||||||||||
41 | OSA_001203 | XX | 01 | MurC | NC1=NC(NC2=NN(C)C(C(C)(C)C)=C2)=C3C(NN=C3)=N1 | N4-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine | BDEUAKAPFVRQSD-UHFFFAOYSA-N | WYH_TR1-5-1-P | 286.3 | |||||||||||||||||||||||||||||||||||||||||||||
42 | OSA_001204 | XX | 01 | MurC | CC(C)(C)C1=CC(NC2=C3C(NN=C3)=NC(OCCCC)=N2)=NN1C | 6-butoxy-N-(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | YYTTZHUMGWXUCV-UHFFFAOYSA-N | WYH17-X-BP | 343.4 | |||||||||||||||||||||||||||||||||||||||||||||
43 | OSA_001205 | XX | 01 | MurC | WYH_TR6-4-3-P | WYH_TR6-4-3-P | 358.4 | |||||||||||||||||||||||||||||||||||||||||||||||
44 | OSA_001206 | XX | 01 | MurC | WYH_TR6-8-P | WYH_TR6-8-P | ||||||||||||||||||||||||||||||||||||||||||||||||
45 | OSA_001207 | XX | 01 | MurC | WYH22-rac | |||||||||||||||||||||||||||||||||||||||||||||||||
46 | OSA_001208 | XX | 01 | MurC | WYH22-R-GBoc | |||||||||||||||||||||||||||||||||||||||||||||||||
47 | OSA_001209 | XX | 01 | MurC | WYH22-rac-GBoc | |||||||||||||||||||||||||||||||||||||||||||||||||
48 | OSA_001210 | XX | 01 | MurC | WYH32-G | |||||||||||||||||||||||||||||||||||||||||||||||||
49 | OSA_001211 | XX | 01 | MurC | WYH22-R-G | |||||||||||||||||||||||||||||||||||||||||||||||||
50 | OSA_001212 | XX | 01 | MurC | WYH22-rac-G | |||||||||||||||||||||||||||||||||||||||||||||||||
51 | OSA_000001 | MurD | 79.6 | CN1CCN(CC1)c1ccc(cc1)C#N | 4-(4-methylpiperazin-1-yl)benzonitrile | ZSDPKKGOSKXEHN-UHFFFAOYSA-N | Z2856434840 | 201.27 | MURD-x0349 | FragLibrary | In Library | https://github.com/opensourceantibiotics/murligase/wiki/MurD-fragment-screen | ZINC000000236863. | 859595 | 261DF2DE2905A04D3FC95058666494DD | SCHEMBL151261 | 763205 | MCULE-3957797171 | MolPort-000-894-567 | J1.186.427I | DTXSID30354088 | |||||||||||||||||||||||||||||||||
52 | OSA_000002 | MurD | 79.6 | CN1CCN(CC1)C(=O)NC1=CC=C(F)C=C1 | N-(4-fluorophenyl)-4-methylpiperazine-1-carboxamide | MDBPFVSVLGYVCQ-UHFFFAOYSA-N | Z2856434944 | 237.28 | MURD-x0373 | FragLibrary | In Library | https://github.com/opensourceantibiotics/murligase/wiki/MurD-fragment-screen | AWD | ZINC000000386890. | 1467788 | C75AA6C64E59D4D569D5A305E87650A6 | SCHEMBL10053027 | 851986 | MCULE-1085231672 | MolPort-001-889-175 | J153.485H | |||||||||||||||||||||||||||||||||
53 | OSA_000003 | MurD | CC(CO)(CO)NC(=O)Nc1ccccc1 | 3-(1,3-dihydroxy-2-methylpropan-2-yl)-1-phenylurea | NLGYHTMGWVQQIL-UHFFFAOYSA-N | Z57472297 | 224.26 | MURD-x0374 | FragLibrary | In Library | https://github.com/opensourceantibiotics/murligase/wiki/MurD-fragment-screen | AYV | ZINC000000408628 | 659431 | 4056614 | MCULE-1218000011 | ||||||||||||||||||||||||||||||||||||||
54 | OSA_000004 | MurD | 72.4 | CC(C(Nc1cc(C#N)ccc1)=O)C | N-(3-cyanophenyl)-2-methylpropanamide | JWBISRKEEZGPFB-UHFFFAOYSA-N | Z26548083 | 188.23 | MURD-x0378 | FragLibrary | In Library | https://github.com/opensourceantibiotics/murligase/wiki/MurD-fragment-screen | ZINC000009254030 | 31406591 | BFF73936E3D5C2A2195B9E9EB364CAA2 | SCHEMBL4599032 | 16383207 | MCULE-2084722473 | MolPort-004-354-760 | |||||||||||||||||||||||||||||||||||
55 | OSA_000738 | MurD | -22.2 | O=C(C1CCN(C)CC1)NC2=CC=C(F)C=C2 | N-(4-fluorophenyl)-1-methylpiperidine-4-carboxamide | FFVXKXJVYNMPKL-UHFFFAOYSA-N | DMK75-2-A | 236.29 | 95968061 | |||||||||||||||||||||||||||||||||||||||||||||
56 | OSA_000739 | MurD | 24.7 | O=C(C1CCN(C)C1)NC2=CC=C(F)C=C2 | N-(4-fluorophenyl)-1-methylpyrrolidine-3-carboxamide | RLOXACRLJWMWPU-UHFFFAOYSA-N | DMK79-1-A | 222.26 | 110858666 | |||||||||||||||||||||||||||||||||||||||||||||
57 | OSA_000740 | MurD | 22.4 | O=C(C1CCN(C)CC1)NC2=CC=CC=C2 | 1-methyl-N-phenylpiperidine-4-carboxamide | CZZZAQIBVXXNRC-UHFFFAOYSA-N | DMK76-1-A | 218.3 | 23377552 | |||||||||||||||||||||||||||||||||||||||||||||
58 | OSA_000741 | MurD | 136 | CN1CCC(C(NC2=CC=C(Cl)C=C2)=O)CC1 | N-(4-chlorophenyl)-1-methylpiperidine-4-carboxamide | HDVFKDCTFBLIGZ-UHFFFAOYSA-N | DMK90-1-A | 252.74 | 95968063 | |||||||||||||||||||||||||||||||||||||||||||||
59 | OSA_000743 | MurD | 107 | O=C(C1CCN(C)CC1)NC2=CC=C(Cl)C(Cl)=C2 | N-(3,4-dichlorophenyl)-1-methylpiperidine-4-carboxamide | KOCUBRJDCKLJCJ-UHFFFAOYSA-N | DMK101-1-A | 287.18 | 68317877 | |||||||||||||||||||||||||||||||||||||||||||||
60 | OSA_000744 | MurD | 114 | O=C(C1CCN(C)CC1)NC2=CC=CC3=C2C=CC=C3 | 1-methyl-N-(naphthalen-1-yl)piperidine-4-carboxamide | XPWQQCGWCGOQQG-UHFFFAOYSA-N | DMK81-4-A | 268.36 | 99817646 | |||||||||||||||||||||||||||||||||||||||||||||
61 | OSA_000745 | MurD | 71.4 | O=C(C1CCN(C)CC1)NC2=CC=CC(O)=C2 | N-(3-hydroxyphenyl)-1-methylpiperidine-4-carboxamide | XAQXZAPPHDDIRP-UHFFFAOYSA-N | DMK85-2-A | 234.3 | ||||||||||||||||||||||||||||||||||||||||||||||
62 | OSA_000746 | MurD | 29.6 | O=C(C1CCN(C)CC1)NC2=CC=C(O)C=C2 | N-(4-hydroxyphenyl)-1-methylpiperidine-4-carboxamide | YOBBRZGGOJZMSA-UHFFFAOYSA-N | DMK98-1-B | 234.3 | ||||||||||||||||||||||||||||||||||||||||||||||
63 | OSA_000747 | MurD | 103 | CN1CCC(C(NC2=CC=C(OC)C=C2)=O)CC1 | N-(4-methoxyphenyl)-1-methylpiperidine-4-carboxamide | VIDFQXVHRPPTSE-UHFFFAOYSA-N | DMK92-1-A | 248.33 | 95968070 | |||||||||||||||||||||||||||||||||||||||||||||
64 | OSA_000748 | MurD | 126 | OC(C(Br)=C1)=CC=C1NC(C2CCN(C)CC2)=O | N-(3-bromo-4-hydroxyphenyl)-1-methylpiperidine-4-carboxamide | OKUOAWCXQVKURI-UHFFFAOYSA-N | DMK104-1-B | 313.2 | ||||||||||||||||||||||||||||||||||||||||||||||
65 | OSA_000750 | MurD | 133 | O=C(C1CCN(C)CC1)NC2=CC=CC=C2Br | N-(2-bromophenyl)-1-methylpiperidine-4-carboxamide | LKXFVAFVNYONFT-UHFFFAOYSA-N | DMK84-2-A | 297.2 | 60004863 | |||||||||||||||||||||||||||||||||||||||||||||
66 | OSA_000751 | MurD | 39.8 | O=C(C1CCN(C)CC1)NC2=CC=CC(Br)=C2 | N-(3-bromophenyl)-1-methylpiperidine-4-carboxamide | ZQBUUHOVMXBKOP-UHFFFAOYSA-N | DMK83-1-A | 297.2 | 95968089 | |||||||||||||||||||||||||||||||||||||||||||||
67 | OSA_000752 | MurD | 78.9 | O=C(C1CCN(C)CC1)NC2=CC=C(Br)C=C2 | N-(4-bromophenyl)-1-methylpiperidine-4-carboxamide | MPGBNJKPYBAROJ-UHFFFAOYSA-N | DMK82-1-A | 297.2 | 51103985 | |||||||||||||||||||||||||||||||||||||||||||||
68 | OSA_000753 | MurD | 41.8 | O=C(C1CCN(C)CC1)NC2=C(C3=CC=CC=C3)C=CC=C2 | N-([1,1'-biphenyl]-2-yl)-1-methylpiperidine-4-carboxamide | WSIROINKJIPLSC-UHFFFAOYSA-N | DMK102-1-A | 294.4 | 99817647 | |||||||||||||||||||||||||||||||||||||||||||||
69 | OSA_000755 | MurD | 15.3 | O=C(C1CCN(C)CC1)NC2=CC=CC(C3=CC=CC=C3)=C2 | N-([1,1'-biphenyl]-3-yl)-1-methylpiperidine-4-carboxamide | DPBBCALZTLCOIT-UHFFFAOYSA-N | DMK87-1-B | 294.4 | ||||||||||||||||||||||||||||||||||||||||||||||
70 | OSA_000756 | MurD | 91.9 | O=C(C1CCN(C)CC1)NC2=CC(C3=CC=C(C=CC=C4)C4=C3)=CC=C2 | 1-methyl-N-(3-(naphthalen-2-yl)phenyl)piperidine-4-carboxamide | RXYMXPPTPPPTLC-UHFFFAOYSA-N | DMK95-1-A | 344.46 | ||||||||||||||||||||||||||||||||||||||||||||||
71 | OSA_000757 | MurD | 35.7 | O=C(C1CCN(C)CC1)NC2=CC=C(C3=CC=CC=C3)C=C2 | N-([1,1'-biphenyl]-4-yl)-1-methylpiperidine-4-carboxamide | GMNHICLLRMPJFX-UHFFFAOYSA-N | DMK96-1-A | 294.4 | ||||||||||||||||||||||||||||||||||||||||||||||
72 | OSA_000758 | MurD | 6.53 | O=C(C1CCN(C)CC1)NC2=CC=C(C3=CC=C(C=CC=C4)C4=C3)C=C2 | 1-methyl-N-(4-(naphthalen-2-yl)phenyl)piperidine-4-carboxamide | HEUZCVPUMTWLAE-UHFFFAOYSA-N | DMK97-1-A | 344.46 | ||||||||||||||||||||||||||||||||||||||||||||||
73 | OSA_000759 | MurD | 13.5 & MurE | O=C(C1CCN(C)CC1)NC2=CC=C(C3=CC=NC=C3)C=C2 | 1-methyl-N-(4-(pyridin-4-yl)phenyl)piperidine-4-carboxamide | FOYCAWNDFDSDPG-UHFFFAOYSA-N | DMK109-1-B | 295.39 | ||||||||||||||||||||||||||||||||||||||||||||||
74 | OSA_000760 | MurD | 106 | O=C(C1CCN(C)CC1)NC2=CC=C(C3=CC=CN=C3)C=C2 | 1-methyl-N-(4-(pyridin-3-yl)phenyl)piperidine-4-carboxamide | VHOFAYQMUVOETF-UHFFFAOYSA-N | DMK110-1-B | 295.39 | ||||||||||||||||||||||||||||||||||||||||||||||
75 | OSA_000761 | MurD | 116 | O=C(C1CCN(C)CC1)NC2=CC(N3CCCCC3)=CC=C2 | 1-methyl-N-(3-(piperidin-1-yl)phenyl)piperidine-4-carboxamide | OXEGRJXFVBEBTB-UHFFFAOYSA-N | DMK89-2-B | 301.43 | ||||||||||||||||||||||||||||||||||||||||||||||
76 | OSA_000762 | MurD | 62.7 | O=C(C1CCN(C)CC1)NC2=CC=C(N3CCOCC3)C=C2 | 1-methyl-N-(4-morpholinophenyl)piperidine-4-carboxamide | GLGKAWALSIJYHG-UHFFFAOYSA-N | DMK112-1-A | 303.41 | ||||||||||||||||||||||||||||||||||||||||||||||
77 | OSA_000763 | MurD | 97.8 | O=C(C1CCN(C)CC1)NC2=CC=C(N3CCCCC3)C=C2 | 1-methyl-N-(4-(piperidin-1-yl)phenyl)piperidine-4-carboxamide | YPWJBXOPAVZHPZ-UHFFFAOYSA-N | DMK106-1-A | 301.43 | 110693529 | |||||||||||||||||||||||||||||||||||||||||||||
78 | OSA_000764 | MurD | 99.6 | O=C(NC1=CC(NC2CCCCC2)=CC=C1)C3CCN(CC3)C | N-(3-(cyclohexylamino)phenyl)-1-methylpiperidine-4-carboxamide | GWOGEIVUIJEMAY-UHFFFAOYSA-N | DMK93-2-A | 315.46 | ||||||||||||||||||||||||||||||||||||||||||||||
79 | OSA_000765 | MurD | 21.2 | O=C(C1CCN(C)CC1)NC2=CC=C(NC(C)C)C=C2 | N-(4-(isopropylamino)phenyl)-1-methylpiperidine-4-carboxamide | VZJYHKRIBTXZAO-UHFFFAOYSA-N | DMK111-1-A | 275.4 | ||||||||||||||||||||||||||||||||||||||||||||||
80 | OSA_000766 | MurD | 92.4 | O=C(C1CCN(C)CC1)NC2=CC=C(NC3CCCCC3)C=C2 | N-(4-(cyclohexylamino)phenyl)-1-methylpiperidine-4-carboxamide | RSFQSAYEJQVTHE-UHFFFAOYSA-N | DMK105-1-A | 315.46 | ||||||||||||||||||||||||||||||||||||||||||||||
81 | OSA_000767 | MurD | 51.3 | CC(C)C1N(C)CCC2=C1NC3=CC=CC=C32 | 1-Isopropyl-2-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole | XIGXNSOZHWZZMB-UHFFFAOYSA-N | FI112-2 | 228.338 | ||||||||||||||||||||||||||||||||||||||||||||||
82 | OSA_000768 | MurD | 197 | BrC1=CC(NC(C)=O)=CC=C1 | N-(3-bromophenyl)acetamide | XXHOHJTVFUJJMT-UHFFFAOYSA-N | FI124-1 | 214.062 | ||||||||||||||||||||||||||||||||||||||||||||||
83 | OSA_000769 | MurD | 203 | O=S(C1=CC=C(NC(C)=O)C=C1)(N2CCN(C3=NC=CC=C3)CC2)=O | N-(4-((4-(pyridin-2-yl)piperazin-1-yl)sulfonyl)phenyl)acetamide | BYKOGXKIENOVFN-UHFFFAOYSA-N | FI130-1 | 360.437 | ||||||||||||||||||||||||||||||||||||||||||||||
84 | OSA_000770 | MurD | 47.8 | O=C(C(C)C)NC1=CC=CC(C2=CN=CC=C2)=C1 | N-(3-(pyridin-3-yl)phenyl)isobutyramide | KWNNCPXCTWFGPN-UHFFFAOYSA-N | FI131-1 | 240.305 | ||||||||||||||||||||||||||||||||||||||||||||||
85 | OSA_000771 | MurD | 29.8 | O=C(C(C)C)NC1=CC=CC(C2=CN=CC=C2)=C1 | 1-Methyl-4-(4-(pyridin-3-yl)phenyl)piperazine | KWNNCPXCTWFGPN-UHFFFAOYSA-N | FI132-1 | 240.305 | ||||||||||||||||||||||||||||||||||||||||||||||
86 | OSA_000772 | MurD | 37.7 | O=S(C1=CC=C(NC(C)=O)C=C1)(N2CCOCC2)=O | N-(4-(Morpholinosulfonyl)phenyl)acetamide | WSVGZFWJCRPWAG-UHFFFAOYSA-N | FI133-1 | 284.335 | ||||||||||||||||||||||||||||||||||||||||||||||
87 | OSA_000773 | MurD | 19.5 | O=S(C1=CC=C(NC(C)=O)C=C1)(NCC2=CC=C(OCO3)C3=C2)=O | N-(4-(N-(benzo[d][1,3]dioxol-5-ylmethyl)sulfamoyl)phenyl)acetamide | QIEXJUZBFRBKML-UHFFFAOYSA-N | FI134-1 | 348.378 | ||||||||||||||||||||||||||||||||||||||||||||||
88 | OSA_000774 | MurD | 35.7 | O=S(C1=CC=C(NC(C)=O)C=C1)(N2CCN(C)CC2)=O | N-(4-((4-methylpiperazin-1-yl)sulfonyl)phenyl)acetamide | FIFVSQIZNIIPJZ-UHFFFAOYSA-N | FI135-1 | 297.378 | ||||||||||||||||||||||||||||||||||||||||||||||
89 | OSA_000775 | MurD | 82.5 | O=S(C1=CC=C(NC(C)=O)C=C1)(NCCN2CCOCC2)=O | N-(4-(N-(2-morpholinoethyl)sulfamoyl)phenyl)acetamide | ACDMONYKERYXRY-UHFFFAOYSA-N | FI136-1 | 327.404 | ||||||||||||||||||||||||||||||||||||||||||||||
90 | OSA_000776 | MurD | 22.2 | O=C(C(C)C)NC1=CC=CC(C2=CC=C(OC3=CC=CC=C3)C=C2)=C1 | N-(4'-phenoxy-[1,1'-biphenyl]-3-yl)isobutyramide | DNPIDTVUKHZLJL-UHFFFAOYSA-N | FI137-1B | 331.414 | ||||||||||||||||||||||||||||||||||||||||||||||
91 | OSA_000777 | MurD | -214 | O=C(C(C)C)NC1=CC=CC(C2=CC=C(OC)C=C2)=C1 | N-(4'-methoxy-[1,1'-biphenyl]-3-yl)isobutyramide | BZSTUXKJLYWJSW-UHFFFAOYSA-N | FI138-1 | 269.343 | ||||||||||||||||||||||||||||||||||||||||||||||
92 | OSA_000778 | MurD | 68.4 | O=S(C1=CC=C(NC(C)=O)C=C1)(N2CCC(O)CC2)=O | N-(4-((4-hydroxypiperidin-1-yl)sulfonyl)phenyl)acetamide | PRLOWNAGHFFGCK-UHFFFAOYSA-N | FI139-1 | 298.362 | ||||||||||||||||||||||||||||||||||||||||||||||
93 | OSA_000779 | MurD | 0 | COC(C=C1)=CC=C1C2=CC=C(N3CCN(C)CC3)C=C2 | 1-(4'-Methoxy-[1,1'-biphenyl]-4-yl)-4-methylpiperazine | SHOSXLCUJJBWML-UHFFFAOYSA-N | FI143-1B | 282.386 | ||||||||||||||||||||||||||||||||||||||||||||||
94 | OSA_000780 | MurD | -9.69 | CN(CC1)CCN1C2=CC=C(C3=CC=C(C=CC=C4)C4=C3)C=C2 | 1-Methyl-4-(4-(naphthalen-2-yl)phenyl)piperazine | CVHJZYYHFDIULT-UHFFFAOYSA-N | FI144-1D | 302.42 | ||||||||||||||||||||||||||||||||||||||||||||||
95 | OSA_000781 | MurD | -531 | O=S(C1=CC=C(NC(C)=O)C=C1)(N2CCN(C3=CC=C(OC)C=C3)CC2)=O | N-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)acetamide | RANNSMVPRJINCO-UHFFFAOYSA-N | FI145-1 | 389.475 | ||||||||||||||||||||||||||||||||||||||||||||||
96 | OSA_000782 | MurD | 101 | O=S(C1=CC=C(NC(C)=O)C=C1)(N2CCN(CCN(C)C)CC2)=O | N-(4-((4-(2-(Dimethylamino)ethyl)piperazin-1-yl)sulfonyl)phenyl)acetamide | PNNHPJSMKNRYIO-UHFFFAOYSA-N | FI146-1 | 354.473 | ||||||||||||||||||||||||||||||||||||||||||||||
97 | OSA_000783 | MurD | 33.6 | O=C(C(C)C)NC1=CC=C(Br)C=C1 | N-(4-bromophenyl)isobutyramide | AVQYIQZFJLEKGK-UHFFFAOYSA-N | FI148-1 | 242.115 | ||||||||||||||||||||||||||||||||||||||||||||||
98 | OSA_000784 | MurD | 0 | CN(CC1)CCN1C2=CC=C(C3=CC=C(OC4=CC=CC=C4)C=C3)C=C2 | 1-Methyl-4-(4'-phenoxy-[1,1'-biphenyl]-4-yl)piperazine | CAAVQSSQPMCJAJ-UHFFFAOYSA-N | FI150-1B | 344.457 | ||||||||||||||||||||||||||||||||||||||||||||||
99 | OSA_000785 | MurD | 149 | O=C(C(C)C)NC1=CC=CC(C2=CC=C(C=CC=C3)C3=C2)=C1 | N-(3-(naphthalen-2-yl)phenyl)isobutyramide | NOXBYDYDGIBFQX-UHFFFAOYSA-N | FI151-1 | 289.377 | ||||||||||||||||||||||||||||||||||||||||||||||
100 | OSA_000786 | MurD | 0.74 | O=C(C(C)C)NC1=CC=CC(C2=CSC3=C2C=CC=C3)=C1 | N-(3-(benzo[b]thiophen-3-yl)phenyl)isobutyramide | RQWZQOIAPNFGGO-UHFFFAOYSA-N | FI152-1 | 295.405 | ||||||||||||||||||||||||||||||||||||||||||||||
101 | OSA_000787 | MurD | -45.8 | O=C(C(C)C)NC1=CC=C(C2=CC=C(C=CC=C3)C3=C2)C=C1 | N-(4-(naphthalen-2-yl)phenyl)isobutyramide | UTCQQWMTVBBWSV-UHFFFAOYSA-N | FI153-1 | 289.377 | ||||||||||||||||||||||||||||||||||||||||||||||
102 | OSA_000789 | MurD | 16.3 & MurE | O=C(C(C)C)NC1=CC=C(C2=CN=CC=C2)C=C1 | N-(4-(pyridin-3-yl)phenyl)isobutyramide | LKTDNYDXCXAMKT-UHFFFAOYSA-N | FI155-1 | 240.305 | ||||||||||||||||||||||||||||||||||||||||||||||
103 | OSA_000790 | MurD | 0 | CN(CC1)CCN1C2=CC=C(C3=CSC4=C3C=CC=C4)C=C2 | 1-(4-(Benzo[b]thiophen-3-yl)phenyl)-4-methylpiperazine | BMJKSOJJPUHDMI-UHFFFAOYSA-N | FI156-1B | 308.448 | ||||||||||||||||||||||||||||||||||||||||||||||
104 | OSA_000791 | MurD | -22.8 | O=C(C(C)C)NC1=CC=C(OC2=CC=C(Cl)C=C2)C=C1 | N-(4-(4-chlorophenoxy)phenyl)isobutyramide | MJRRKYUCTQTSAN-UHFFFAOYSA-N | FI157-1 | 289.761 | ||||||||||||||||||||||||||||||||||||||||||||||
105 | OSA_000792 | MurD | 931 | O=C(C(C)C)NC1=CC=C(C2=CC=C(OC)C=C2)C=C1 | N-(4'-methoxy-[1,1'-biphenyl]-4-yl)isobutyramide | GCEQZQIQTAMELE-UHFFFAOYSA-N | FI158-1 | 269.343 | ||||||||||||||||||||||||||||||||||||||||||||||
106 | OSA_000793 | MurD | 255 | O=C(C(C)C)NC1=CC=C(C2=CC=C(OC3=CC=CC=C3)C=C2)C=C1 | N-(4'-phenoxy-[1,1'-biphenyl]-4-yl)isobutyramide | AXKLEVSJVNZWNQ-UHFFFAOYSA-N | FI159-1 | 331.414 | ||||||||||||||||||||||||||||||||||||||||||||||
107 | OSA_000794 | MurD | 78.7 | O=C(C(C)C)NC1=CC=C(OC2=CC=C(Cl)C=C2)C(Cl)=C1 | N-(3-chloro-4-(4-chlorophenoxy)phenyl)isobutyramide | BYQIARDUTWTXAZ-UHFFFAOYSA-N | FI160-1 | 324.206 | ||||||||||||||||||||||||||||||||||||||||||||||
108 | OSA_000795 | MurD | 60.4 | O=C(C(C)C)NC1=CC=C(CN2N=CN=C2)C=C1 | N-(4-((1H-1,2,4-triazol-1-yl)methyl)phenyl)isobutyramide | SVTQNBMLUNRJJH-UHFFFAOYSA-N | FI161-1 | 244.297 | ||||||||||||||||||||||||||||||||||||||||||||||
109 | OSA_000796 | MurD | 11.5 | O=C(C(C)C)NC1=CC=C(C2=CC=C(OC)C(O)=C2)C=C1 | N-(3'-Hydroxy-4'-methoxy-[1,1'-biphenyl]-4-yl)isobutyramide | DKWPQKAHBKWPKB-UHFFFAOYSA-N | FI162-1A | 285.342 | ||||||||||||||||||||||||||||||||||||||||||||||
110 | OSA_000797 | MurD | 70.3 | CN(CC1)CCN1C2=CC=C(NC(C3=CC=CO3)=O)C=C2 | N-(4-(4-methylpiperazin-1-yl)phenyl)furan-2-carboxamide | ZFNBQDCDCYWTTO-UHFFFAOYSA-N | FI163-1 | 285.346 |