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Treatment of corneal and periocular neoplasia in horses: beyond the scalpel

Izak Venter

+27 833089237

izak@vetsfocus.co.za

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Ocular neoplasia

Most common ocular tumors in the horse:

  • Squamous cell carcinomas
  • Sarcoid
  • Melanomas

10% of all equine neoplasms

Locally invasive with a risk of recurrence

Anatomical location:

Orbit

Eyelids/palpebral conjunctiva

Third eyelid

Cornea/sclera/bulbar conjunctiva

Intraocular

Therapeutic challenges

  • Majority of equine ocular neoplasms are malignant (locally invasive with a risk of recurrence)
  • Complete excision with margins is often impossible

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Adnexal neoplasia

Common

Squamous cell carcinoma [SCC]

Sarcoid

 Uncommon

Papilloma

Melanoma

Lymphosarcoma

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Corneal neoplasia

Common

Squamous cell carcinoma [SCC]

Very Uncommon

Papilloma

Melanoma

Haemangioma

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Squamous cell carcinoma [SCC]

Mucocutaneous squamous cell carcinoma (MC-SCC)

  • Second most common skin tumour
  • Second most common equine tumour overall

The nature of MC-SCC varies widely

Slow growing, benign tumours

Rapidly growing, highly malignant and invasive tumours

Frequency of metastasis for MC-SCC is reported to be as high as 19%

Local lymph nodes

Salivary glands

Lungs

Unilateral disease is typical

Bilateral involvement can be as high as 20%

Examine contralateral, ‘unaffected’ eye

Serosanguinous ocular discharge

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Pathogenesis

Chronic irritation

  • Neoplastic transformation of epithelium into SCC

UV radiation

  • High elevations
  • Light hair and minimal skin pigmentation
  • p53 mutation

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Pathogenesis

Equine caballus papillomavirus-2 (EcPV-2)

  • 100% of ocular SCC lesions
  • 50% of ocular swabs from healthy horses

Necessary but not sufficient

UV drives most periocular SCC, while EcPV-2 is a major oncogenic initiator

Both converge through COX-mediated tumour progression

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Pathogenesis

🌞 Chronic UV Exposure (Initiation)

⬇�• UV-B DNA damage

• Reactive oxygen species (ROS)�• Local immunosuppression

🧬 Genetic Damage & Mutation

⬇�• p53 mutation → ↓ apoptosis�• DNA repair failure�• Clonal expansion of mutated keratinocytes

🔬 Pre-Neoplastic Change

⬇�Hyperplasia → Dysplasia → Carcinoma in situ

🔥 COX-2 Upregulation (Occurs early after UV exposure. )

⬇�↑ COX-2 → ↑ Prostaglandin E2 (PGE2)

Effects:

  • ↑ Cell proliferation
  • ↓ Apoptosis
  • ↑ Angiogenesis (↑ VEGF)
  • ↑ Invasion (↑ MMPs)
  • ↓ Immune surveillance

🧫 Invasive Squamous Cell Carcinoma

⬇�• Basement membrane invasion�• Local tissue destruction�• ± Regional metastasis

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Clinical signs

Small superficial nodules

Covered with normal skin

Ulceration and malodorous necrosis

Hyperemic eyelid erosive plaques

Papillomatous SCC

Raised mass with a pink, cobblestone appearance

Ulceration

Necrosis

Infiltrate the orbit

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Clinical signs

Small superficial nodules

Covered with normal skin

Ulceration and malodorous necrosis

Hyperemic eyelid erosive plaques

Papillomatous SCC

Raised mass with a pink, cobblestone appearance

Ulceration

Necrosis

Infiltrate the orbit

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Differential diagnosis

  • Equine sarcoid
  • Habronemiasis
  • Cutaneous lymphoma

  • Melanoma
  • Papilloma
  • Mast cell tumour
  • Exuberant granulation tissue
  • Phycomycosis

Habronema

Calcified material

Cytology - eosinophils

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Diagnosis

Local lymph nodes palpation and fine needle aspirates

Biopsy and histopathology

  • G1 (grade 1)
    • Well-differentiated tumours
  • G3 (grade 3)
    • Poorly differentiated
    • Anaplastic squamous cells
    • High nuclear : cytoplasmic ratio
    • Mitotic figures
  • Grade 2 (G2)
    • Moderately differentiated

Metastasis

44% for G3

3% for G1

25% for G2 

80 % G3 tumours

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Treatment SCC

Surgical management

Cryotherapy

Hyperthermia

Radiotherapy

Chemotherapy

Photodynamic therapy

Most successful when treatment is initiated early

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Surgical treatment

Visible tumour = tip of iceberg

Beyond margins:

UV-damaged epithelium

Mutated keratinocyte clones

COX-driven inflammatory microenvironment

± Viral oncogenesis contribution

Microscopic disease remains after “complete excision”

If you only remove what you can see, you leave behind what caused it

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Surgical treatment

Debulk total tumor size

2‐cm tumor‐free margin

  • Impossible in most cases

Extensive blepharoplastic procedures

  • Facial skin is firmly attached
  • Poor superficial blood supply
  • No “excess” skin

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Surgical treatment

Enucleation/exenteration

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Cryotherapy �

Liquid nitrogen at -196°C

Lyse tumour cells - intracellular ice formation

Double or triple freeze–thaw cycle

Rapid freeze and slow thaw

Protect the underlying cornea

Early or precancerous SCC

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Radiotherapy�

Ionising radiation

Damage nucleic acids and protein

Free radical formation

  • Teletherapy
    • Multiple treatments
    • General anaesthesia
    • Not practical
  • Brachytherapy

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Brachytherapy

Gamma radioactive sources

High dose of radiation

Minimal radiation to surrounding tissues

Isotopes

  • Gold, radon, cesium, and tantalum Iridium

Parallel rows approximately 1 cm apart

Total treatment time 7 days

High cost, limited availability, licensure issues, and human radiation exposure

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Anti-neoplastic Pharmacologic Classification

Cytotoxics

Mechanism: Direct tumour cell kill or replication inhibition

Examples:

  • Intratumoural cisplatin
  • Mitomycin C
  • 5-fluorouracil (5-FU)
  • Bleomycin

�➡ Direct DNA damage or replication interference�➡ True cytotoxic pharmacology

Immune-Mediated Anti-Neoplastic Agents (Non-Classical Cytostatics)

Mechanism: Immune activation → tumour control

Examples:

  • Imiquimod

�➡ TLR-7 immune activation�➡ Indirect tumour suppression

NSAIDs with Anti-Neoplastic Activity (Adjunct Tumour Modulation)

Mechanism: COX inhibition → ↓ PGE2 → tumour microenvironment effects

Examples:

  • Piroxicam

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Cisplatin

Inhibits DNA synthesis by binding to DNA

Intralesional injection

10 mg/ml, followed by mixing with sesame seed oil (60%)

3.3 mg cisplatin/ml

1 mg cisplatin/cm3 of tissue

4 intra tumoral injections given at 2-week intervals

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Cisplatin implants

Cisplatin-containing biodegradable pellets [1.6 mg, 3 mg]

Localized, sustained-release chemotherapy

Each bead releases cisplatin over approximately 4–5 weeks, achieving high local cytotoxic concentrations while minimizing systemic exposure and toxicity

Advantages

  • Safer handling
  • Consistent intralesional distribution
  • Fewer treatment sessions than intralesional cisplatin oil

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Cisplatin implants

Lesion Type / Location

Recommended Bead Strength

Rationale

Periocular, eyelid, lip, nasal regions

1.6 mg

Reliable release profile and tissue penetration without corneal irritation

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Cisplatin implants

Tumour Bed

Area (cm²)

No. of 1.6 mg Beads

Total Dose (mg)

3 × 3 cm

9

3

4.8

4 × 3 cm

12

4

6.4

6 × 5 cm

30

10

16

Dosage and Placement

  • Each bead diffuses active drug to approximately a 1 cm radius
  • Spacing: Place beads 1.5 cm apart within and just beyond the tumour margins

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Cisplatin implants

Tumour Type

Long-term Resolution (≥ 2 years)

Notes

Sarcoid & spindle-cell tumours

≈ 91 %

High remission

Minimal adverse effects

Squamous cell carcinoma (SCC)

60–83 %

Best results with debulking + beads

Melanoma

≈ 93 %

Durable response, especially in grey horses

Clinical Efficacy

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Cisplatin implants

Adverse Effects

• Mild transient local inflammation or oedema

• Keratitis risk if implanted too close to cornea or upper eyelid

• Systemic absorption minimal

Post-operative Management

• NSAID: Flunixin 1.1 mg/kg PO q24 h × 3 days

• Advise handlers to avoid contact with wound exudate due to residual cisplatin risk

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Imiquimod: Clinical Pharmacology�

Immune Response Enhancement

Interferon-α (IFN-α)

TNF

IL-8, 10, 12

TLR-7 / 8 → NF-κB → Cytokine burst

Drives both innate and adaptive anti-tumour immune responses

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Imiquimod

Cellular Immune Effects

Innate Immune Activation

  • Recruitment of plasmacytoid dendritic cells (PDCs)
  • High local Type I interferon production

Antigen Presentation Enhancement

  • Maturation of epidermal Langerhans cells
  • Migration to regional lymph nodes

Adaptive Immune Activation

  • Antigen-specific cytotoxic T-cell activation
  • Enhanced tumour immune recognition

Skin application� ↓�Dendritic cell activation� ↓�Lymph node priming� ↓�Cytotoxic T-cell tumour targeting

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Direct Tumour Microenvironment Effects

Pro-Apoptotic Effects

  • ↑ Death receptors (CD95 / Fas)
  • ↓ Anti-apoptotic proteins (Bcl-2)

Anti-Angiogenic Effects

  • IFN-α
  • IL-10
  • IL-12
  • MMP inhibitors

  • bFGF
  • MMP-9

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Imiquimod

DOSAGE AND ADMINISTRATION:

Apply three times weekly

More frequent application does not enhance therapeutic outcomes and may exacerbate local irritation.

Treatment duration typically ranges from 2 to 3 months for small lesions.

SIDE EFFECTS:

Erythema

Alopecia

Exudation

Depigmentation

Typically emerge within two weeks

Subside within 8 weeks

NB Pro inflammatory product

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Mitomycin C

Antineoplastic antibiotic (Streptomyces caespitosus )

Bioreductive alkylating agent

Potent cytotoxic effect on rapidly dividing cells

Inhibits fibrosis and wound healing responses

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Mechanism of Action

�MMC = DNA Damage + Anti-Fibrotic = Dual Anti-Tumour Effect

�DNA cross-linking� ↓�Inhibits DNA synthesis � ↓�Tumour cell apoptosis / necrosis

PLUS

↓ Fibroblast proliferation�↓ ECM production�↓ Post-surgical scarring

MMC basically locks tumour DNA closed — if DNA can’t open, the tumour can’t grow

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Why MMC Works Well for Ocular SCC

Treats entire ocular surface → hits subclinical disease

Can reduce recurrence vs surgery alone

Can be used: Alone / Post-debulking

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Indications

Primary Corneal SCC

Limbal SCC

Third eyelid SCC

Conjunctival SCC

Best use scenarios

  • Small–moderate lesions
  • Residual microscopic disease post surgery
  • Owners declining surgery

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Dosage Protocol

Typical protocol

  • 0.04% solution~1–2 drops q6h 7 days ON → 7 days OFF
  • Up to 4 cycles
  • Week-on / week-off protects limbal stem cells

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Evidence Snapshot

Equine study outcomes

MMC alone → resolution in 6 / 8 eyes

Surgery + MMC → resolution in 7 / 9 eyes

No major complications reported

Shows favourable comparison to surgery alone recurrence rates

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COX inhibition: Piroxicam�

Not a primary curative therapy

Adjunct / supportive anti-tumour therapy

SCC often has inflammatory + COX-2 driven biology

Piroxicam = COX inhibition → potential anti-tumour effect

COX-2–derived prostaglandins are linked to tumour growth, angiogenesis and metastasis

COX inhibition →

↓ Prostaglandin E2 →

↓ Tumour cell survival signals

↓ Angiogenesis

↓ Immunosuppression

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�Equine Sarcoid

Locally invasive

Benign fibroblastic skin tumours

Most common equine tumour

Key Concepts

  • Inactive sarcoids may become aggressive after injury, biopsy or inappropriate treatment.
  • Major functional + cosmetic impact
  • Do not metastasize
  • an be clinically aggressive

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�Classification�

Aggression ↑ → Need multimodal therapy

Low aggression

High aggression

Ocult

Fibroblastic

Verrucous

Mixed

Nodular

Malevolant

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�Aetiology

Core Drivers

  • BPV 1 & 2 infection
  • Genetic susceptibility
  • Trauma / wounds
  • Possible fly vector transmission

BPV is causally associated with sarcoid development, but infection alone is not sufficient.

Flies may act as mechanical vectors

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�Treatment

Why Are There 40+ Treatments?”

Because no single treatment works for all sarcoids

There is no consistently reliable treatment for every sarcoid type, location and patient.

What desperation + internet advice produces

Burnt toast rubbed on lesion

Cigarette ash paste

Toothpaste + baking soda mixtures

Superglue “to suffocate tumour”

Battery acid

Household bleach

Vinegar soaks

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�Diagnosis

Presumptive diagnosis based on

clinical appearance

Presence of more than one lesion with characteristics of sarcoid is strongly suggestive

Definitive diagnosis - histopathology

Biopsy-induced trauma or irritation may exacerbate the lesion and induce proliferation

Biopsy ONLY if treatment planned immediately

Never wake the dragon unless you are ready to kill it

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Treatment

Not All Sarcoids React The Same

Options include:

  • Surgery
  • Cisplatin (implant or injection)
  • 5-FU
  • Imiquimod
  • BCG
  • Radiation
  • Cryotherapy
  • Electrochemotherapy
  • AW5: Fluorouracil, thiouracil, heavy metal salts, and steroid

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�Treatment

🚫 High-Risk “Do Not Cut First” Sarcoids

Periocular Sarcoids

  • High recurrence
  • Functional risk (eyelid damage)

Fibroblastic / Ulcerated Sarcoids

  • Highly reactive
  • Trauma → explosive growth

Previously Interfered Sarcoids

  • Surgery / ligation / caustics history
  • Often biologically “activated”

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�Treatment

🚫 High-Risk “Do Not Cut First” Sarcoids

Periocular Sarcoids

  • High recurrence
  • Functional risk (eyelid damage)

Fibroblastic / Ulcerated Sarcoids

  • Highly reactive
  • Trauma → explosive growth

Previously Interfered Sarcoids

  • Surgery / ligation / caustics history
  • Often biologically “activated”

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Periocular oncology is unforgiving

Small decisions create permanent outcomes

Precision matters more than aggression

Think first

Cut last